Search Results
- SY-690693 - 690693 AKT1, AKT2, AKT3 Kinase Inhibitor
- AKT1, AKT2, AKT3 inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- SY-A769662 - A769662 AMPK Kinase Inhibitor
- AMPK inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- SY-ABT-737 - ABT-737 Bcl-2 Kinase Inhibitor
- Bcl-2 inhibitor. Inquire for pricing on 5, 10, 50, 100 mg sizes. ... More
- SY-ABT-869 - ABT-869 (796967-16-3) Multi Kinase Inhibitor
- Multi Kinase Inhibitor (Flt3, PDGFR & VEGFR) (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-AKT-I-1 - AKt-I-1 AKT Kinase Inhibitor
- AKT inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes) ... More
- SY-AMG-Tie2 - AMG-Tie2 TIE-2 Kinase Inhibitor
- TIE-2 inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-AT-7519 - AT-7519 CDK Kinase Inhibitor
- CDK inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-AV951 - AV951 VEGF Kinase Inhibitor
- VEGF inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-AZ-960 - AZ-960 JAKs Kinase Inhibitor
- JAKs inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- SY-AZD6244 - AZD6244 MEK Kinase Inhibitor
- MEK inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-AZD7762 - AZD7762 CHK Kinase Inhibitor
- CHK inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- PKI-ADPHTN-005 - Adaphostin
- Adaphostin is a lipophilic, adamantyl ester of BCR-ABL tyrosine kinase inhibitor tyrphostin AG 957, purity: > 97% (HPLC) ... More
- SY-AKT-I-1,2 - Akt-I-1,2 AKT Kinase Inhibitor
- AKT inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes) ... More
- PKI-AKT-005 - Akt1/2 Inhibitor
- isozyme selective Akt1/2 kinase inhibitor, noncompetitive with ATP, purity: > 98% (HPLC) ... More
- PKI-AMGT-005 - Aminogenistein
- Aminogenistein is a Lck tyrosine kinase inhibitor, purity: > 98% (HPLC) ... More
- SY-Axitinib - Axitinib (AG013736) Multi Kinase Inhibitor (cKIT, PDGFR & VEGFR)
- Multi Kinase Inhibitor (cKIT, PDGFR & VEGFR) (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-BI-2536R - BI-2536(R-) PLK Kinase Inhibitor
- PLK inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-BI-D1870 - BI-D1870 RSK Kinase Inhibitor
- RSK inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-BMS-2 - BMS-2 MET Kinase Inhibitor
- MET inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-BX795 - BX795 PDK1/TBK1 Kinase Inhibitor
- PDK1/TBK1 inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-BX912 - BX912 PDK1 Kinase Inhibitor
- PDK1 inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-Bosutinib - Bosutinib Multi Kinase Inhibitor
- Multi Kinase Inhibitor (Abl , Src) inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- SY-CC-401 - CC-401 JNK Kinase Inhibitor
- JNK inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- SY-CHIR-258 - CHIR-258 Multi Kinase Inhibitor
- Multi Kinase Inhibitor (c-Kit,FGFR, FLT3,FMS,PDGFR, VEGFR) inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- SY-CI-1040 - CI-1040 MEK Kinase Inhibitor
- MEK inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- SY-CP-690550 - CP-690550 JAKs Kinase Inhibitor
- JAKs inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-CP-724714 - CP-724714 ErbB2 Kinase Inhibitor
- ErbB2 inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-Canertinib - Canertinib, CI-1033 EGFR Kinase Inhibitor
- EGFR inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-Dasatinib - Dasatinib Multi Kinase Inhibitor (Bcr-Abl, EAR, c-Kit & PDGFR)
- Multi Kinase Inhibitor (Bcr-Abl, EAR, c-Kit & PDGFR) (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-E7080 - E7080 Multi Kinase Inhibitor (VEGF, FGF & SCF)
- Multi Kinase Inhibitor (VEGF, FGF & SCF) (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- IAP002 - Easy 50 PI3K Inhibitor Array
- Isoform-specific inhibitors of proteins in the PI3 kinase (PI3K) signalling pathway prepared in a convenient, easy-to-use 96-well plate format. Assays with the complete panel of inhibitors enable you to dissect which specific signaling pathway m ... More
- SY-Erlotinib - Erlotinib EGFR Kinase Inhibitor
- EGFR inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-Flavopiridol - Flavopiridol (Alvocidib, HMR-1275) CDK Kinase Inhibitor
- CDK inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-GDC-0941 - GDC-0941 (957054-30-7) PI3K Kinase Inhibitor
- PI3K inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- PKI-GW5074-010 - GW 5074
- GW 5074 is a selective and cell-permeable c-Raf (Raf1) kinase inhibitor, purity: > 98% (HPLC) ... More
- SY-GW441756 - GW441756 TrkA Kinase Inhibitor
- TrkA inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-Gefitinib - Gefitinib EGFR Kinase Inhibitor
- EGFR inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- PKI-GFTB2-200 - Gefitinib Purity: 99,0 percent
- Gefitinib, or IRESSATM as it is more commonly called, is an epidermal growth factor receptor tyrosine kinase inhibitor (EGFR-TKI). EGFR is part of the ERBB receptor family, which has four closely related members: EGFR (ERBB1), HER2 (ERBB2), HER3 (ERB ... More
- PKI-GFTB2-050 - Gefitinib Purity: 99,0 percent
- Gefitinib, or IRESSATM as it is more commonly called, is an epidermal growth factor receptor tyrosine kinase inhibitor (EGFR-TKI). EGFR is part of the ERBB receptor family, which has four closely related members: EGFR (ERBB1), HER2 (ERBB2), HER3 (ERB ... More
- PKI-GFTB2-010 - Gefitinib Purity: 99.0 percent
- Gefitinib is a potent and specific EGFR tyrosine kinase inhibitor, purity: > 99.0% (HPLC) ... More
- PKI-GFTB-010 - Gefitinib Purity: 99.9 percent
- Gefitinib is a potent and specific EGFR tyrosine kinase inhibitor, purity: > 99.9% (HPLC) ... More
- PKI-HOFAS-005 - Hydroxyfasudil
- Hydroxyfasudil is a Rho kinase inhibitor, active metabolite of fasudil (HA-1077), purity: > 98% (HPLC) ... More
- SY-IC87114 - IC87114 PI3K Kinase Inhibitor
- PI3K inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- PKI-IMTB-010 - Imatinib Mesylate
- Imatinib, formerly referred to as STI571, is a specific Bcr-Abl tyrosine kinase inhibitor, purity: 99% (HPLC) ... More
- SY-Imatinib - Imatinib mesylate BCR-ABL Kinase Inhibitor
- BCR-ABL inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-JNJ38877605 - JNJ38877605 MET Kinase Inhibitor
- MET inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- SY-JNJ7706621 - JNJ7706621 AUR (CDK) Kinase Inhibitor
- AUR (CDK) inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-KU0063794 - KU0063794 mTOR Kinase Inhibitor
- mTOR inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-KU55933 - KU55933 ATM Kinase Inhibitor
- ATM inhibitor (inquire about pricing for 5, 10, 50, and 100 mg sizes) ... More
- SY-Ki20227 - Ki20227 FMS Kinase Inhibitor
- FMS inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-AP24534 - Kinase Inhibitor - AP24534
- AP24534 is active against pan-BCR-ABL (IC50=0.37nM) and mutated form (IC50=0.3-2.0nM), VEGFR2(IC50=1.5nM), FGFR1(IC50=2.2nM), PDGFR (IC50=1.1nM) and LYN (IC50=0.24nM). AP24534, a Pan-BCR-ABL Inhibitor for Chronic Myeloid Leukemia, Potently Inhibits t ... More
- SY-Lapatinib - Lapatinib EGFR; HER2 Kinase Inhibitor
- EGFR; HER2 inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- SY-MP-470 - MP-470 AUR Kinase Inhibitor
- AUR inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-Masatinib - Masatinib c-Kit Kinase Inhibitor
- c-Kit inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- SY-Mk-5 - Mk-5 JAKs Kinase Inhibitor
- JAKs inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- SY-Motesanib - Motesanib Multi Kinase Inhibitor (c-Kit, PDGFR & VEGFR)
- Multi Kinase Inhibitor (c-Kit, PDGFR & VEGFR) (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-Nilotinib - Nilotinib Multi Kinase Inhibitor (Bcr-Abl, Kit & PDGFR)
- Multi Kinase Inhibitor (Bcr-Abl, Kit & PDGFR) (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-TPL2Kinhib - Other Kinase Inhibitor - Tpl2 Kinase Inhibitor
- A cell-permeable, potent, reversible, and ATP-competitive inhibitor of Tpl2 kinase (IC50 = 50 nM). Please inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- PKI-PD169-001 - PD 169316
- PD 169316 is a potent and cell-permeable p38 MAP kinase inhibitor, purity: > 98% (HPLC) ... More
- SY-PD0325901 - PD0325901 MEK Kinase Inhibitor
- MEK inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-PD-04217903 - PD04217903 MET Kinase Inhibitor
- MET inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- SY-PD173955 - PD173955 BCR-ABL Kinase Inhibitor
- BCR-ABL inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- SY-D-64406 - PDGF-R PTK Inhibitor - PDGFR tyrosine Kinase Inhibitor I
- A cell-permeable bis (1H-2-indolyl)-1-methanone compound that acts as a highly selective, ATP-competitive, and reversible inhibitor of platelet-derived growth factor (PDGF) receptor tyrosine kinase (IC50 = 200 nM in Swiss 3T3 cells for PDGFR; IC50 = ... More
- SY-PF562271 - PF-562271 FAK; RTKs Kinase Inhibitor
- FAK; RTKs inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- SY-PF431396 - PF431396 PYK2 Kinase Inhibitor
- PYK2 inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-PI-103 - PI103 PI3K Kinase Inhibitor
- PI3K inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- SY-PIK-93 - PIK93 PI3K Kinase Inhibitor
- PI3K inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- PKA-PKI-100 - PKI, heat-stable protein kinase inhibitor of PKA
- PKI is a recombinant heat-stable protein kinase inhibitor PKI (full length, ... More
- PKA-PKI-500 - PKI, heat-stable protein kinase inhibitor of PKA (rabbit)
- The heatstable protein kinase inhibitor PKI is a key role player for the regulation of PKA activity and for localizing the catalytic subunit of PKAin the cell, also working as a nuclear scavenger. This relatively small protein (77 amino acids) is ext ... More
- SY-PLX4720 - PLX4720 RAF Kinase Inhibitor
- RAF inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-KRN633 - PTK Inhibitor - VEGFR Tyrosine Kinase Inhibitor III, KRN633
- A cell-permeable, reversible, ATP-competitive inhibitor of VEGFR kinase activity (IC50 = 170 nM, 160 nM, and 125 nM for VEGFR-1, VEGFR-2, VEGFR-3, respectively). Inhibits PDGFR-a and c-Kit only at higher concentrations (IC50 = 0.97 uM and 4.33 uM, re ... More
- SY-Pazopanib - Pazopanib VEGFR Kinase Inhibitor
- VEGFR inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- PKI-PCTL-010 - Piceatannol
- Piceatannol is a Syk/ZAP70-specific kinase inhibitor, purity: > 98% (HPLC) ... More
- SY-AG957 - Protein Tyrosine Kinase (PTK) Inhibitor - AG957
- A potent tyrosine kinase inhibitor. Selectively blocks the tyrosine kinase activity of human p210bcr-abl (Ki = 750 nM) over p140c-abl (Ki = 10 uM). Please inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- SY-Purvalanol B - Purvalanol B CDK Kinase Inhibitor
- CDK inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- SY-RHO-15 - RHO-15 RHO Kinase Inhibitor
- RHO inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-H1152P - Rho Kinase Inhibitor
- A cell-permeable isoquinolinesulfonamide compound that acts as a highly specific, reversible, potent, and ATP-competitive inhibitor of G-protein Rho-associated kinase (ROCK; Ki = 1.6 nM). Exhibits a much weaker affinity for other serine/threonine kin ... More
- SY-SB-216763 - SB-216763 GSK 3 Kinase Inhibitor
- GSK 3 inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- SY-SB-202190 - SB202190 (152121-30-7) MAPK (p38MAP) Kinase Inhibitor
- MAPK (p38MAP) inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- SY-SB-203580 - SB203580 (152121-47-6) MAPK (p38MAP) Kinase Inhibitor
- MAPK (p38MAP) inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- SY-SB590885 - SB590885 B-Raf Kinase Inhibitor
- B-Raf inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-SD169 - SD169 p38 MAPK Kinase Inhibitor
- p38 MAPK inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- SY-SNS-032 - SNS-032 CDK Kinase Inhibitor
- CDK inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-SNS-314 - SNS-314 Aurora Kinase Inhibitor
- Aurora inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-SR3677 - SR3677 PROCK-II Kinase Inhibitor
- PROCK-II (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- PKI-SU11274-001 - SU11274
- SU 11274 is a Met tyrosine kinase inhibitor, purity: > 98% (HPLC) ... More
- SY-SU-5402 - SU5402 c-Kit Kinase Inhibitor
- c-Kit inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- PKI-SU6656-005 - SU6656
- SU 6656 is a potent src family kinase inhibitor and inhibits Src (IC50 = 280 nM) as well as closely related kinases such as Fyn (IC50 = 170 nM), Yes (IC50 = 20 nM) and Lyn (IC50 = 130 nM). Inhibition is competitive to ATP. It acts as a weak inhibitor ... More
- PKI-SU6656-001 - SU6656
- SU 6656 is a potent src family kinase inhibitor and inhibits SRC, FYN, YES and LYN, purity: > 98% (HPLC) ... More
- PKI-POLYPHEN-500 - Set of polyphenolic compounds
- Polyphenolic compounds are especially food constituents of plant origin comprising a variety of phenolic structures. The main classes of polyphenols are defined according to the nature of their carbon skeleton: flavonoids, phenolic acids, phenolic al ... More
- SY-Sorafenib - Sorafenib Multi Kinase Inhibitor (B-Raf & VEGFR)
- Multi Kinase Inhibitor (B-Raf & VEGFR) (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-4PDiMQ - Src Family PTK Inhibitor - Src Kinase Inhibitor I
- A potent, selective, dual site, cell-permeable, reversible and ATP-competitive inhibitor of Src family tyrosine kinases (IC50 = 44 nM and 88 nM for Src and Lck, respectively). Shown to simultaneously interact with both the ATP- and peptide-binding si ... More
- SY-567806 - Src Family PTK Inhibitor - Src Kinase Inhibitor II
- A potent, ATP-competitive, reversible and selective inhibitor of Src family tyrosine kinases (IC50 = 1.2 �M for human recombinant Csk). Please inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- 6212 - Staurosporine
- Staurosporine, isolated from Streptomyces sp., is a protein kinase inhibitor. Staurosporine induces DNA fragmentation and apoptosis at 1mM in 2-3 hours. ... More
- SY-Sunitinib - Sunitinib Multi Kinase Inhibitor (CSF-1R, Flt3, Kit, PDGFR, RET & VEGFR)
- Multi Kinase Inhibitor (CSF-1R, Flt3, Kit, PDGFR, RET & VEGFR) (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-TGX221 - TGX-221 PI3K Kinase Inhibitor
- PI3K inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- SY-Tandutinib - Tandutinib (CT53518, MLN518) Multi Kinase Inhibitor (cKIT, Flt3, PDGFR)
- Multi Kinase Inhibitor (cKIT, Flt3, PDGFR) (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-AC220 - Tyrosine Kinase Inhibitor - AC220
- AC220 is a novel, orally available, small molecule that has been optimized as a selective FMS-like tyrosine kinase-3 (FLT3) inhibitor. It is currently in clinical development for the treatment of AML ... More
- PKI-AG490-010 - Tyrphostin AG 490
- Tyrphostin AG 490 is a potent JAK-2 protein tyrosine kinase inhibitor and also inhibits EGFR tyrosine kinase, purity: > 98% (HPLC) ... More
- PKI-AG490-025 - Tyrphostin AG 490
- Tyrphostin AG 490 is a specific and potent JAK-2 protein tyrosine kinase inhibitor and also inhibits EGF receptor autophosphorylation, with an IC50 of 100 nM. It inhibits DNA synthesis and cell growth and induces apoptosis. Photosensitive. ... More
- SY-VEGFRTKV - VEGF-R PTK Inhibitor - VEGFR Tyrosine Kinase Inhibitor V
- A cell-permeable, ATP-binding pocket-targeting N-cyclopropylnaphthamide compound that acts as a potent inhibitor against VEGFR1/2/3 (IC50 = 0.6 nM against VEGFR2), c-FMS, RET, Lyn, and c-KIt, while exhibiting much reduced activity against 36 other co ... More
- SY-VX-680 - VX-680 AUR Kinase Inhibitor
- AUR inhibitor (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-VX-702 - VX-702 (479543-46-9) MAPK (p38MAP) Kinase Inhibitor
- MAPK (p38MAP) inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes) ... More
- SY-Vandetanib - Vandetanib EGFR, VEGFR Kinase Inhibitor
- EGFR, VEGFR inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- SY-Vargatef - Vargatef Multi Kinase Inhibitor (VEGF, FGFR & SCF)
- Multi Kinase Inhibitor (VEGF, FGFR & SCF) (inquire for pricing on 5, 10, 50, 100 mg sizes) ... More
- SY-YM201636 - YM201636 PIKfyve Kinase Inhibitor
- PIKfyve inhibitor (inquire about pricing for 5mg, 10mg, 50mg, and 100mg sizes ... More
- SY-XL880 - cMET Inhibitor - XL880
- XL880 is a novel MET and VEGFR2 kinase inhibitor with an IC50 of 0.4 and 0.8 nM for MET and VEGFR2, respectively ... More